論文・総説 - 細谷　孝充

101. Kanemoto K, Yoshida S, Hosoya T. Modified Conditions for Copper-Catalyzed ipso-Thiolation of Arylboronic Acid Esters with Thiosulfonates. Chem Lett. 2018.01; 47 (1): 85-88. ( DOI )

102. Kusuhara H, Takashima T, Fujii H, Takashima T, Tanaka M, Ishii A, Tazawa S, Takahashi K, Takahashi K, Tokai H, Yano T, Kataoka M, Inano A, Yoshida S, Hosoya T, Sugiyama Y, Yamashita S, Hojo T, Watanabe Y. Comparison of pharmacokinetics of newly discovered aromatase inhibitors by a cassette microdosing approach in healthy Japanese subjects. Drug Metab Pharmacokinet. 2017.12; 32 (6): 293-300. ( PubMed, DOI )

103. Yoshida S, Shimizu K, Uchida K, Hazama Y, Igawa K, Tomooka K, Hosoya T. Construction of Condensed Polycyclic Aromatic Frameworks through Intramolecular Cycloaddition Reactions Involving Arynes Bearing an Internal Alkyne Moiety. Chem Eur J. 2017.11; 23 (61): 15332-15335. ( PubMed, DOI )

104. Matsuzawa T, Uchida K, Yoshida S, Hosoya T. Synthesis of Diverse o-Arylthio-Substituted Diaryl Ethers by Direct Oxythiolation of Arynes with Diaryl Sulfoxides Involving Migratory O-Arylation. Org Lett. 2017.10; 19 (20): 5521-5524. ( PubMed, DOI )

105. Hatakeyama M, Sakamoto Y, Ogata K, Sumida Y, Sumida T, Hosoya T, Nakamura S. A study on an unusual S_N2 mechanism in the methylation of benzyne through nickel-complexation. Phys Chem Chem Phys. 2017.10; 19 (39): 26926-26933. ( PubMed, DOI )

106. Nakano-Kobayashi A, Awaya T, Kii I, Sumida Y, Okuno Y, Yoshida S, Sumida T, Inoue H, Hosoya T, Hagiwara M. Prenatal neurogenesis induction therapy normalizes brain structure and function in Down syndrome mice. Proc Natl Acad Sci USA. 2017.09; 114 (38): 10268-10273. ( PubMed, DOI )

107. Kanemoto K, Sugimura Y, Shimizu S, Yoshida S, Hosoya T. Rhodium-catalyzed odorless synthesis of diaryl sulfides from borylarenes and S-aryl thiosulfonates. Chem Commun. 2017.09; 53 (77): 10640-10643. ( PubMed, DOI )

108. Sakaguchi H, Uetake Y, Ohashi M, Niwa T, Ogoshi S, Hosoya T. Copper-Catalyzed Regioselective Monodefluoroborylation of Polyfluoroalkenes en Route to Diverse Fluoroalkenes. J Am Chem Soc. 2017.09; 139 (36): 12855-12862. ( PubMed, DOI )

109. Niwa T, Ochiai H, Hosoya T. Facile Transformation of α,β-Unsaturated Carboxylic Acids to Alkenylboronic Esters via Rhodium-Catalyzed Decarbonylative Borylation of α,β-Unsaturated Thioesters. Chem Lett. 2017.09; 46 (9): 1315-1318. ( DOI )

110. Meguro T, Yoshida S, Hosoya T. Sequential Molecular Conjugation using Thiophene S,S-Dioxides Bearing a Clickable Functional Group. Chem Lett. 2017.08; 46 (8): 1137-1140. ( DOI )

111. Nishiyama Y, Hazama Y, Yoshida S, Hosoya T. Synthesis of Unsymmetrical Tertiary Phosphine Oxides via Sequential Substitution Reaction of Phosphonic Acid Dithioesters with Grignard Reagents. Org Lett. 2017.07; 19 (14): 3899-3902. ( PubMed, DOI )

112. Furubayashi T, Motohashi K, Wakao K, Matsuda T, Kii I, Hosoya T, Hayashi N, Sadaie M, Ishikawa F, Matsushita M, Fujiyoshi S. Three-Dimensional Localization of an Individual Fluorescent Molecule with Angstrom Precision. J Am Chem Soc. 2017.07; 139 (26): 8990-8994. ( PubMed, DOI )

113. Nakamura Y, Yoshida S, Hosoya T. Facile Synthesis of Phthalides from Methyl ortho-Iodobenzoates and Ketones via an Iodine–Magnesium Exchange Reaction Using a Silylmethyl Grignard Reagent. Chem Lett. 2017.06; 46 (6): 858-861. ( DOI )

114. Sumida Y, Sumida T, Hosoya T. Nickel-Catalyzed Reductive Cross-Coupling of Aryl Triflates and Nonaflates with Alkyl Iodides. Synthesis. 2017.06; 49 (16): 3590-3601. ( DOI )

115. Yoshida S, Nagai A, Uchida K, Hosoya T. Enhancing the Synthetic Utility of 3-Haloaryne Intermediates by their Efficient Generation from Readily Synthesizable ortho-Iodoaryl Triflate-type Precursors. Chem Lett. 2017.05; 46 (5): 733-736. ( DOI )

116. Niwa T, Ochia H, Hosoya T. Copper-Catalyzed ipso-Borylation of Fluoroarenes. ACS Catal. 2017.05; 7 (7): 4535-4541. ( DOI )

117. Sako Y, Ninomiya K, Okuno Y, Toyomoto M, Nishida A, Koike Y, Ohe K, Kii I, Yoshida S, Hashimoto N, Hosoya T, Matsuo M, Hagiwara M. Development of an orally available inhibitor of CLK1 for skipping a mutated dystrophin exon in Duchenne muscular dystrophy. Sci Rep. 2017.05; 7 46126. ( PubMed, DOI )

118. Meguro T, Yoshida S, Hosoya T . Aromatic Azido-selective Reduction via the Staudinger Reaction Using Tri-n-butylphosphonium Tetrafluoroborate with Triethylamine. Chem Lett. 2017.04; 46 (4): 473-476. ( DOI )

119. Uchida K, Yoshida S, Hosoya T. Three-Component Coupling of Triflyloxy-Substituted Benzocyclobutenones, Organolithium Reagents, and Arynophiles Promoted by Generation of Aryne via Carbon-Carbon Bond Cleavage. Org Lett. 2017.03; 19 (5): 1184-1187. ( PubMed, DOI )

120. Ochiai H, Uetake Y, Niwa T, Hosoya T. Rhodium-Catalyzed Decarbonylative Borylation of Aromatic Thioesters for Facile Diversification of Aromatic Carboxylic Acids. Angew Chem Int Ed. 2017.02; 56 (9): 2482-2486. ( PubMed, DOI )