論文・総説 - 細谷　孝充

21. Miyazaki Y, Kikuchi M, Umezawa K, Descamps A, Nakamura D, Furuie G, Sumida T, Saito K, Kimura N, Niwa T, Sumida Y, Umehara T, Hosoya T, Kii I. Structure-activity relationship for the folding intermediate-selective inhibition of DYRK1A. Eur J Med Chem. 2022.01; 227 113948. ( PubMed, DOI )

22. Inouye S, Nakamura M, Hosoya T. Enzymatic conversion of dehydrocoelenterazine to coelenterazine using FMN-bound flavin reductase of NAD(P)H:FMN oxidoreductase. Biochem Biophys Res Commun. 2022.01; 587 24-28. ( PubMed, DOI )

23. Niwa T, Uetake Y, Isoda M, Takimoto T, Nakaoka M, Hashizume D, Sakurai H, Hosoya T. Lewis acid-mediated Suzuki–Miyaura cross-coupling reaction. Nat Catal. 2021.12; 4 (12): 1080-1088. ( DOI )

24. Inouye S, Nakamura M, Hosoya T. Formation of Coelenteramine from 2-Peroxycoelenterazine in the Ca²⁺-Binding Photoprotein Aequorin. Photochem Photobiol. 2021.12; ( PubMed, DOI )

25. Takahashi K, Hosoya T, Onoe K, Mori T, Tazawa S, Mawatari A, Wada Y, Watanabe Y, Doi H, Watanabe Y. PET imaging of brain aromatase in humans and rhesus monkeys by ¹¹C-labeled cetrozole analogs. Sci Rep. 2021.12; 11 (1): 23623. ( PubMed, DOI )

26. Sakata Y, Yoshida S, Hosoya T. Synthesis of Azidoanilines by the Buchwald-Hartwig Amination. J Org Chem. 2021.11; 86 (21): 15674-15688. ( PubMed, DOI )

27. Taguchi J, Kimura K, Igawa K, Tomooka K, Hosoya T. 3-Azidoarynes: Generation and Regioselective Reactions. Chem Lett. 2021.11; 51 (2): 94-98. ( DOI )

28. Watanabe K, Terao N, Niwa T, Hosoya T. Direct 3-Acylation of Indolizines by Carboxylic Acids for the Practical Synthesis of Red Light-Releasable Caged Carboxylic Acids. J Org Chem. 2021.09; 86 (17): 11822-11834. ( PubMed, DOI )

29. Inouye S, Sumida Y, Tomabechi Y, Taguchi J, Shirouzu M, Hosoya T. Chiral deaza-coelenterazine analogs for probing a substrate-binding site in the Ca²⁺-binding photoprotein aequorin. PLoS ONE. 2021.06; 16 (6): e0251743. ( PubMed, DOI )

30. Kobayashi K, Matsuzawa T, Hosoya T, Yoshida S. Thioxanthone Synthesis from Benzoic Acid Esters through Directed ortho-Lithiation. Chem Lett. 2021.06; 50 (9): 1624-1627. ( DOI )

31. Aimi T, Meguro T, Kobayashi A, Hosoya T, Yoshida S. Nucleophilic transformations of azido-containing carbonyl compounds via protection of the azido group. Chem Commun. 2021.06; 57 (49): 6062-6065. ( PubMed, DOI )

32. Yoshida S, Hosoya T. Recent Insertion Reactions of Aryne Intermediates. Modern Aryne Chemistry (Ed. Biju AT). 2021.05; 111-148. ( DOI )

33. Kobayashi T, Hosoya T, Yoshida S. Facile Synthetic Methods for Diverse N-Arylphenylalanine Derivatives via Transformations of Aryne Intermediates and Cross-Coupling Reactions. Bull Chem Soc Jpn. 2021.05; 94 (7): 1823-1832. ( DOI )

34. Matsuzawa T, Hosoya T, Yoshida S. Transition-Metal-Free Synthesis of N-Arylphenothiazines through an N- and S-Arylation Sequence. Org Lett. 2021.03; 23 (6): 2347-2352. ( PubMed, DOI )

35. Minoshima M, Uchida K, Nakamura Y, Hosoya T, Yoshida S. Acylalkylation of Arynes Generated from o-Iodoaryl Triflates with Hydrosilanes and Cesium Fluoride. Org Lett. 2021.03; 23 (5): 1868-1873. ( PubMed, DOI )

36. Nakajima H, Hazama Y, Sakata Y, Uchida K, Hosoya T, Yoshida S. Diverse diaryl sulfide synthesis through consecutive aryne reactions. Chem Commun. 2021.03; 57 (21): 2621-2624. ( PubMed, DOI )

37. Suzuki M, Kanemoto K, Nakamura Y, Hosoya T, Yoshida S. Palladium-Catalyzed Sulfinylation of Aryl- and Alkenylborons with Sulfinate Esters. Org Lett. 2021.03; 23 (9): 3793-3797. ( PubMed, DOI )

38. Toyomoto M, Inoue A, Iida K, Denawa M, Kii I, Kadj F M N, Kishi T, Im D, Shimamura T, Onogi H, Yoshida S, Iwata S, Aoki J, Hosoya T, Hagiwara M. S1PR3–G₁₂-biased agonist ALESIA targets cancer metabolism and promotes glucose starvation. Cell Chem Biol. 2021.02; 28 (8): 1132-1144. ( PubMed, DOI )

39. Isoda M, Uetake Y, Takimoto T, Tsuda J, Hosoya T, Niwa T. Convergent Synthesis of Fluoroalkenes Using a Dual-Reactive Unit. J Org Chem. 2021.01; 86 (2): 1622-1632. ( PubMed, DOI )

40. Yoshida S, Sakata Y, Misawa Y, Morita T, Kuribara T, Ito H, Koike Y, Kii I, Hosoya T. Assembly of four modules onto a tetraazide platform by consecutive 1,2,3-triazole formations. Chem Commun. 2021.01; 57 (7): 899-902. ( PubMed, DOI )